academic article

• (Het)aryl Difluoromethyl-Substituted β-Alkoxyenones: Synthesis and Heterocyclizations 2020
• 3-Carboxy-/3-Aminobicyclo[1.1.1]pentane-Derived Sulfonamides and Sulfonyl Fluorides - Advanced Bifunctional Reagents for Organic Synthesis and Drug Discovery 2020
• gem -Difluorocyclopropanation of Alkenyl Trifluoroborates with the CF ₃ SiMe ₃ -NaI System 2020
• Aliphatic α-Boryl-α-bromoketones: Synthesis and Reactivity 2020
• Cycloadditions of Alkenylboronic Derivatives 2020
• Cyclopropyl boronic derivatives in parallel synthesis of sp3-enriched compound libraries 2020
• Fluoroalkyl-Substituted Cyclopropane Derivatives: Synthesis and Physicochemical Properties 2020
• Formyl MIDA Boronate: C ₁ Building Block Enables Straightforward Access to α‐Functionalized Organoboron Derivatives 2020
• Formyl MIDA Boronate: C ₁ Building Block Enables Straightforward Access to α‐Functionalized Organoboron Derivatives 2020
• Front Cover: (Het)aryl Difluoromethyl-Substituted β-Alkoxyenones: Synthesis and Heterocyclizations (Eur. J. Org. Chem. /2020) 2020
• Front Cover: Aliphatic α-Boryl-α-bromoketones: Synthesis and Reactivity (Eur. J. Org. Chem. 23/2020) 2020
• Frontispiece: The Symbiotic Relationship Between Drug Discovery and Organic Chemistry 2020
• Functionalization of 2-Trifluoromethyl-1 H -pyrrole: A Convenient Entry into Advanced Fluorinated Building Blocks Including all Isomeric 2-(Trifluoromethyl)prolines 2020
• Generating Multibillion Chemical Space of Readily Accessible Screening Compounds 2020
• Photochemical [2 + 2] Cycloaddition of Alkenyl Boronic Derivatives: An Entry into 3-Azabicyclo[3.2.0]heptane Scaffold 2020
• Saturated Bicyclic Sultams 2020
• Synthesis of Fused Pyridine Carboxylates by Reaction of β-Alkoxyvinyl Glyoxylates with Amino Heterocycles 2020
• Synthesis of Spirocyclic β- and γ-Sultams by One-Pot Reductive Cyclization of Cyanoalkylsulfonyl Fluorides 2020
• Synthesis of saturated nitrogen heterocycles by Strecker reaction – nucleophilic cyclization 2020
• Twisting and Turning the Sulfonamide Bond: A Synthetic, Quantum Chemical, and Crystallographic Study 2020
• Last of the -Difluorocycloalkanes: Synthesis and Characterization of 2,2-Difluorocyclobutyl-Substituted Building Blocks 2019
• 2,2-Difluorovinyl Pinacolborane - A New Versatile Reagent for the Suzuki-Miyaura Reaction 2019
• N -Difluorocyclopropyl-Substituted Pyrazoles: Synthesis and Reactivity 2019
• Far Away from Flatland. Synthesis and Molecular Structure of Dihetera[3.3. n ]propellanes and Trihetera[3.3. n ]propellanes: Advanced Analogues of Morpholine/Piperazine 2019
• Formation of 10/12/14-Membered Rings is Favored over 5/6/7-Membered. An Unexpected Result from Oxazole Chemistry 2019
• Front Cover: N -Difluorocyclopropyl-Substituted Pyrazoles: Synthesis and Reactivity (Eur. J. Org. Chem. 27/2019) 2019
• Front Cover: Scalable and Straightforward Synthesis of All Isomeric (Cyclo)alkylpiperidines (Eur. J. Org. Chem. 23/2019) 2019
• Front Cover: Sulfonimidamides and Imidosulfuric Diamides: Compounds from an Underexplored Part of Biologically Relevant Chemical Space (Chem. Eur. J. 28/2019) 2019
• Front Cover: Widely Exploited, Yet Unreported: Regiocontrolled Synthesis and the Suzuki-Miyaura Reactions of Bromooxazole Building Blocks (Eur. J. Org. Chem. 18/2019) 2019
• Multigram Synthesis of Functionalized Spirocyclic Diazirines 2019
• One-Pot Parallel Synthesis of 5-(Dialkylamino)tetrazoles 2019
• Regioselective Synthesis of Functionalized 3- or 5-Fluoroalkyl Isoxazoles and Pyrazoles from Fluoroalkyl Ynones and Binucleophiles 2019
• Robust and Scalable Approach to 1,3-Disubstituted Pyridylcyclobutanes 2019
• SAR by Space: Enriching Hit Sets from the Chemical Space 2019
• Scalable Synthesis of Biologically Relevant Spirocyclic Pyrrolidines 2019
• Scalable and Straightforward Synthesis of All Isomeric (Cyclo)alkylpiperidines 2019
• Sulfonimidamides and Imidosulfuric Diamides: Compounds from an Underexplored Part of Biologically Relevant Chemical Space 2019
• Sulfonimidamides and Imidosulfuric Diamides: Compounds from an Underexplored Part of Biologically Relevant Chemical Space 2019
• Synthesis of 1-hetaryl-2,2-difluorocyclopropane-derived building blocks: The case of pyrazoles 2019
• The Boron-Wittig Olefination of Aldehydes and Ketones with Bis[(pinacolato)boryl]methane: an Extended Reaction Scope 2019
• The Symbiotic Relationship Between Drug Discovery and Organic Chemistry 2019
• Widely Exploited, Yet Unreported: Regiocontrolled Synthesis and the Suzuki-Miyaura Reactions of Bromooxazole Building Blocks 2019
• Regioselective synthesis of isoxazole and 1,2,4-oxadiazole-derived phosphonates [3 + 2] cycloaddition 2018
• (Chlorosulfonyl)benzenesulfonyl Fluorides—Versatile Building Blocks for Combinatorial Chemistry: Design, Synthesis and Evaluation of a Covalent Inhibitor Library 2018
• 3-((Hetera)cyclobutyl)azetidines, “Stretched” Analogues of Piperidine, Piperazine, and Morpholine: Advanced Building Blocks for Drug Discovery 2018
• Cover Feature: Synthesis of Bi- and Polyfunctional Isoxazoles from Amino Acid Derived Halogenoximes and Active Methylene Nitriles (Eur. J. Org. Chem. 22/2018) 2018
• Following Ramachandran 2: exit vector plot (EVP) analysis of disubstituted saturated rings 2018
• Hetaryl Bromides Bearing the SO ₂ F Group - Versatile Substrates for Palladium-Catalyzed C-C Coupling Reactions 2018
• Straightforward hit identification approach in fragment-based discovery of bromodomain-containing protein 4 (BRD4) inhibitors 2018
• Synthesis of 3-Azabicyclo[3.2.0]heptane-Derived Building Blocks via [3+2] Cycloaddition 2018
• Synthesis of 4-Hetarylisoxazoles from Amino Acid-Derived Halogenoximes and Push-Pull Enamines 2018
• Synthesis of Bi- and Polyfunctional Isoxazoles from Amino Acid Derived Halogenoximes and Active Methylene Nitriles 2018
• [3+2] Cycloaddition of an Azomethyne Ylide and Vinyl Sulfonyl Fluorides ― an Approach to Pyrrolidine-3-sulfonyl Fluorides 2018